Numerion Labs Funding, Investors & Competitors

Numerion Labs has raised $239M across 6 funding rounds, most recently a $20M Series D in March 2026.

Last Numerion Labs funding round

$20M

Series D · Mar 2026

Cumulative funding Numerion Labs raised

$239M

across 6 funding rounds

Key investors in Numerion Labs

  • Y Combinator
  • DCVC
  • Khosla Ventures
  • Tencent
  • B Capital
  • AME Cloud Ventures
  • Threshold
  • Baidu Ventures

Numerion Labs Overview

About Numerion Labs

Numerion Labs is a preclinical pharmaceutical company using AtomNet deep learning for structure-based drug discovery. The platform targets over 600 unique disease areas, including undruggable proteins, in partnership with more than 250 pharmaceutical, biotech, and agrochemical firms worldwide. Advancing small-molecule candidates into preclinical studies, Numerion Labs operates from the United States with significant venture backing.


Founded

2012

HQ

United StatesSan Francisco, CA

Status

Privately held

Customer focus

B2B

Revenue model

Licensing

Numerion Labs Funding History

Numerion Labs has raised a total of $239M across 6 funding rounds.

Numerion Labs' first fundraising round was a $100K pre-seed round in March 2015. The most recent completed round was a $20M Series D in March 2026.

Numerion Labs funding rounds

Numerion Labs funding rounds
DateStageInvestorsRaised
Mar 2026Series D-$20M
Jan 2024Series C-$45M
Aug 2020Series BB Capital (lead); Sanabil (lead); Y Combinator; Tencent; AME Cloud Ventures; Colorcon; Baidu Ventures; Cerity Partners Ventures; Dolby Family Ventures; DCVC$123M
Mar 2018Series AMonsanto Growth Ventures (MGV) (lead); Y Combinator; Tencent; Baidu Ventures; Khosla Ventures; Dolby Family Ventures; DCVC; B Capital; Threshold$45M
Jun 2015SeedAME Cloud Ventures; Khosla Ventures; Mission and Market; DCVC; Farzad Nazem; OS Fund; Threshold; Draper Associates$6M
Mar 2015Pre-seedY Combinator; David E. Weekly$100K

Who has invested in Numerion Labs?

18 investors have backed Numerion Labs across its funding rounds, including Y Combinator, DCVC, Khosla Ventures, Tencent, B Capital and AME Cloud Ventures.

Lead investors include B Capital, Sanabil and Monsanto Growth Ventures (MGV).


Numerion Labs Investors

Investors in Numerion Labs by funding rounds participated
InvestorHQRoundsRoleFirst check
Y CombinatorUnited StatesSan Francisco, CA3ParticipantMar 2015
DCVCUnited StatesUnited States3ParticipantJun 2015
TencentChinaShenzhen2ParticipantMar 2018
AME Cloud VenturesUnited StatesSan Francisco, CA2ParticipantJun 2015
Baidu VenturesChinaBeijing2ParticipantMar 2018
Khosla VenturesUnited StatesSan Francisco, CA2ParticipantJun 2015
Dolby Family VenturesUnited StatesSan Francisco, CA2ParticipantMar 2018
B CapitalUnited StatesLos Angeles, CA2LeadMar 2018
ThresholdUnited StatesSan Francisco, CA2ParticipantJun 2015
ColorconUnited StatesPhiladelphia, PA1ParticipantAug 2020
Cerity Partners VenturesUnited StatesHaddonfield, NJ1ParticipantAug 2020
Mission and MarketUnited StatesSan Francisco, CA1ParticipantJun 2015
David E. WeeklyUnited StatesSan Francisco, CA1ParticipantMar 2015

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Numerion Labs Competitors

Numerion Labs competitors include listed companies like Merck KGaA and Eli Lilly, and private ones like Astromech, Anew Labs, Sinovac Life Sciences and Intrepid Labs.

Public and private companies comparable to Numerion Labs
CompanyHQStatusRevenueEBITDAValuationRevenue Multiple
AstromechUnited StatesUnited StatesPrivate--$3.8B-
Anew LabsChinaShanghaiPrivate--$1.5B-
Merck KGaAGermanyGermanyPublicly listed$24B$5.3B$66B3.1x
Sinovac Life SciencesChinaBeijingPrivate--$3.3B-
Intrepid LabsCanadaTorontoPrivate--$6.8B-
Eli LillyUnited StatesUnited StatesPublicly listed$65B$28B$1.0T13.1x

Numerion Labs Public Comps

Numerion Labs is still privately-owned, but its public comps include Eli Lilly, Johnson & Johnson, AbbVie, Merck, Roche, Novartis, AstraZeneca, CrowdStrike, SAP and Amgen.

Last FYEV/RevenueEV/EBITDA
RevenueEBITDALast FYLTM2027ELast FYLTM2027E
Eli Lilly$65B$28B16.5x13.1x38.7x27.0x
Johnson & Johnson$94B$40B7.2x6.8x17.0x18.3x
AbbVie$61B$17B8.7x8.1x30.6x17.6x
Merck$65B$28B6.3x6.2x14.7x21.0x
Roche$77B$26B5.0x4.9x14.6x12.4x
Novartis$57B$22B5.5x5.5x14.2x13.3x
AstraZeneca$59B$19B4.8x4.5x14.6x12.7x
CrowdStrike$4.8B($12M)51.4x44.5x(19816.2x)151.0x

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Common questions about Numerion Labs

When was Numerion Labs founded?Numerion Labs was founded in 2012.
Where is Numerion Labs headquartered?Numerion Labs is headquartered in San Francisco, CA, United States.
Is Numerion Labs publicly listed?No, Numerion Labs is a private, VC-backed company.
How much funding has Numerion Labs raised?Numerion Labs has raised $239M across 6 funding rounds.
What was Numerion Labs' last funding round?Numerion Labs' last funding round was a $20M Series D in March 2026.
Who are Numerion Labs' investors?Numerion Labs' investors include Y Combinator, DCVC, Tencent, AME Cloud Ventures, Baidu Ventures, Khosla Ventures, Dolby Family Ventures, B Capital, Threshold, Colorcon and 8 others.
Which companies are comparable to Numerion Labs?Companies comparable to Numerion Labs include Astromech, Anew Labs, Merck KGaA, Sinovac Life Sciences, Intrepid Labs and Eli Lilly.

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